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Chemical Structure : Clobenpropit
Catalog No.: PC-35222Not For Human Use, Lab Use Only.
Clobenpropit (VUF-9153) is a highly potent histamine H3 antagonist/inverse agonist with pA2 value of 9.93, also displays partial agonist activity at H4 receptors.
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Clobenpropit (VUF-9153) is a highly potent histamine H3 antagonist/inverse agonist with pA2 value of 9.93, also displays partial agonist activity at H4 receptors; increases brain histidine decarboxylase activity dose dependently, inhibits electrically induced convulsions in mice.
| M.Wt | 308.828 | |
| Formula | C14H17ClN4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Yokoyama H, et al. Eur J Pharmacol. 1994 Jul 21;260(1):23-8.
2. Clark EA, et al. Br J Pharmacol. 1995 Jan;114(2):357-62.
3. Stark H, et al. J Med Chem. 1996 Mar 1;39(5):1157-63.
4. Mochizuki T, et al. Brain Res. 1996 Dec 16;743(1-2):178-83.
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