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Clobenpropit

Chemical Structure : Clobenpropit

CAS No.: 145231-45-4

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Clobenpropit (VUF-9153, VUF9153)

Catalog No.: PC-35222Not For Human Use, Lab Use Only.

Clobenpropit (VUF-9153) is a highly potent histamine H3 antagonist/inverse agonist with pA2 value of 9.93, also displays partial agonist activity at H4 receptors.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    Clobenpropit (VUF-9153) is a highly potent histamine H3 antagonist/inverse agonist with pA2 value of 9.93, also displays partial agonist activity at H4 receptors.
    Clobenpropit (VUF-9153) increases brain histidine decarboxylase activity dose dependently, inhibits electrically induced convulsions in mice.

    Physicochemical Properties

    M.Wt 308.828
    Formula C14H17ClN4S
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    Carbamimidothioic acid, [(4-chlorophenyl)methyl]-, 3-(1H-imidazol-4-yl)propyl ester (9CI)

    References

    1. Yokoyama H, et al. Eur J Pharmacol. 1994 Jul 21;260(1):23-8.

    2. Clark EA, et al. Br J Pharmacol. 1995 Jan;114(2):357-62.

    3. Stark H, et al. J Med Chem. 1996 Mar 1;39(5):1157-63.

    4. Mochizuki T, et al. Brain Res. 1996 Dec 16;743(1-2):178-83.

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