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Clobenpropit dihydrobromide

Chemical Structure : Clobenpropit dihydrobromide

CAS No.: 145231-35-2

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Clobenpropit dihydrobromide (VUF-9153;VUF9153)

Catalog No.: PC-35223Not For Human Use, Lab Use Only.

Clobenpropit (VUF-9153) is a highly potent histamine H3 antagonist/inverse agonist with pA2 value of 9.93, also displays partial agonist activity at H4 receptors.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Clobenpropit (VUF-9153) is a highly potent histamine H3 antagonist/inverse agonist with pA2 value of 9.93, also displays partial agonist activity at H4 receptors.
Clobenpropit (VUF-9153) increases brain histidine decarboxylase activity dose dependently, inhibits electrically induced convulsions in mice.

Physicochemical Properties

M.Wt 381.744
Formula C14H19Cl3N4S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

3-(1H-imidazol-4-yl)propyl (4-chlorobenzyl)carbamimidothioate dihydrochloride

References

1. Yokoyama H, et al. Eur J Pharmacol. 1994 Jul 21;260(1):23-8.

2. Clark EA, et al. Br J Pharmacol. 1995 Jan;114(2):357-62.

3. Stark H, et al. J Med Chem. 1996 Mar 1;39(5):1157-63.

4. Mochizuki T, et al. Brain Res. 1996 Dec 16;743(1-2):178-83.

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