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Chemical Structure : Conivaptan
CAS No.: 210101-16-9
Catalog No.: PC-70166Not For Human Use, Lab Use Only.
Conivaptan (YM-087) is a potent, selective, nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 25 mg | $248 | In stock | |
| 50 mg | $398 | In stock | |
| 100 mg | $588 | In stock | |
| 200 mg | Get quote | ||
| 1 g | Get quote |
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Conivaptan (YM-087) is a potent, selective, nonpeptide vasopressin V1A and V2 receptor antagonist with Ki of 0.48 nM and 3.04 nM respectively.
Conivaptan (YM-087) has less potency for OT receptors and no effect on V1B receptor.
Conivaptan (YM-087) blocks AVP-induced cAMP production of cultured renal epithelium cells concentration dependently and has no agonistic activities.
| M.Wt | 498.583 | |
| Formula | C32H26N4O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
N-[4-[(4,5-Dihydro-2-methylimidazo[4,5-d][1]benzazepin-6(1H)-yl)carbonyl]phenyl]-[1,1'-Biphenyl]-2-carboxamide |
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1. Tahara A, et al. J Pharmacol Exp Ther. 1997 Jul;282(1):301-8.
2. Tahara A, et al. Cardiovasc Res. 1998 Apr;38(1):198-205.
3. Nakayama S, et al. Neurocrit Care. 2016 Apr;24(2):273-82.
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