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Chemical Structure : Contezolid
CAS No.: 1112968-42-9
Catalog No.: PC-61371Not For Human Use, Lab Use Only.
Contezolid (MRX I) is an orally active oxazolidinone agent with antibacterial activity Gram-positive pathogens, including MRSA, penicillin-PRSP, PISP, and vancomycin-resistant enterococci (VRE) with MIC of 0.25-4 ug/mL.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $388 | In stock | |
| 10 mg | $588 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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Contezolid (MRX I) is an orally active oxazolidinone agent with antibacterial activity Gram-positive pathogens, including MRSA, penicillin-PRSP, PISP, and vancomycin-resistant enterococci (VRE) with MIC of 0.25-4 ug/mL.
Contezolid demonstrates the same or better efficacy than linezolid in both systemic and local infection models against the tested strains.
| M.Wt | 408.337 | |
| Formula | C18H15F3N4O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
1-{2,3,6-trifluoro-4-[(5S)-5-{[(1,2-oxazol-3-yl)amino]methyl}-2-oxo-1,3-oxazolidin-3-yl]phenyl}-2,3-dihydropyridin-4(1H)-one |
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1. Li CR, et al. Antimicrob Agents Chemother. 2014;58(4):2418-21.
2. Gordeev MF, et al. J Med Chem. 2014 Jun 12;57(11):4487-97.
3. Meng J, et al. Drug Metab Dispos. 2015 May;43(5):646-59.
4. Eckburg PB, et al. Antimicrob Agents Chemother. 2017 Mar 24;61(4). pii: e02181-16.
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