Chemical Structure : DAS-CHO-5-oCRBN
CAS No.:
DAS-CHO-5-oCRBN
(c-Src PROTAC degrader)
Catalog No. : PC-21653Not For Human Use, Lab Use Only.
DAS-CHO-5-oCRBN is a potent and selective PROTAC for c-Src kinase with DC50 value of 55 nM in CAL148 cells.
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Purity & Documentation Purity:
98.9% (HPLC) Select Batch: PC-2165301
Biological Activity
DAS-CHO-5-oCRBN is a potent and selective PROTAC for c-Src kinase with DC50 value of 55 nM in CAL148 cells.
Physicochemical Properties
M.Wt
883.99
Formula
C45H45N11O7S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
2-((6-(4-(2-(4-(2-(2,6-dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)piperazin-1-yl)-2-oxoethyl)piperazin-1-yl)-2-methylpyrimidin-4-yl)amino)-N-(2-methyl-4-phenoxyphenyl)thiazole-5-carboxamide
References
1. Mao W, et al. ACS Chem Biol
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