DC-TEADin02

Chemical Structure : DC-TEADin02

CAS No.: 2380228-45-3

Catalog No.: PC-23121Not For Human Use, Lab Use Only.

DC-TEADin02 is a potent, selective, covalent TEAD autopalmitoylation inhibitor with IC50 of 197 nM, shows minimal effect on TEAD-YAP interaction.

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10 mg	$58	In stock
25 mg	$98	In stock
50 mg	$158	In stock
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Biological Activity

DC-TEADin02 is a potent, selective, covalent TEAD autopalmitoylation inhibitor with IC50 of 197 nM, shows minimal effect on TEAD-YAP interaction.
DC-TEADin02 exhibits specific thiol reactivity and selectivity of DC-TEADin02 over the kinase family, lipid-binding proteins and epigenetic targets.
DC-TEADin02 inhibited TEADs transcription activity leading to downregulation of YAP-related downstream gene expression.

Physicochemical Properties

M.Wt	323.41
Formula	C19H17NO2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(4-(Naphthalen-2-ylmethyl)phenyl)ethenesulfonamide

References

1. Lu W, et al. Eur J Med Chem. 2019 Dec 15;184:111767.

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DC-TEADin02

Biological Activity

Physicochemical Properties

References

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