DG013A | ERAP1 inhibitor | Probechem Biochemicals

Chemical Structure : DG013A

CAS No.: 2007955-07-7

DG013A (DG 013A)

Catalog No.: PC-72271Not For Human Use, Lab Use Only.

DG013A (DG 013A) is tripeptide mimetic chemical probe (inhibitor) of ERAP1 with IC50 of 0.19 uM, 15-fold selectivity over ERAP2, potently inhibits aminopeptidase N (APN) with IC50 of 3.7 nM.

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Biological Activity

DG013A (DG 013A) is tripeptide mimetic chemical probe (inhibitor) of ERAP1 with IC50 of 0.19 uM, 15-fold selectivity over ERAP2, potently inhibits aminopeptidase N (APN) with IC50 of 3.7 nM.

Physicochemical Properties

M.Wt	512.591
Formula	C27H37N4O4P
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	((S)-2-(((S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl)carbamoyl)-4-methylpentyl)((R)-1-amino-3-phenylpropyl)phosphinic acid

References

1. Birgit Wilding, et al. Bioorg Med Chem Lett. 2021 Jun 15;42:128050.

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DG013A (DG 013A)

Biological Activity

Physicochemical Properties

References

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