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DPI-287

Chemical Structure : DPI-287

CAS No.: 519058-13-0

DPI-287 (DPI 287)

Catalog No.: PC-49552Not For Human Use, Lab Use Only.

DPI-287 is a small-molecule agonist of the δ-opioid receptor (DOP, DOR) with Ki vaule of 0.39 nM, shows 10-fold selectivity for DOP over MOP (Ki=3.17 nM).

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    DPI-287 is a small-molecule agonist of the δ-opioid receptor (DOP, DOR) with Ki vaule of 0.39 nM, shows 10-fold selectivity for DOP over MOP (Ki=3.17 nM).

    Physicochemical Properties

    M.Wt 485.67
    Formula C31H39N3O2
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    4-((R)-((2S,5R)-4-benzyl-2,5-dimethylpiperazin-1-yl)(3-hydroxyphenyl)methyl)-N,N-diethylbenzamide

    References

    1. Tobias Claff, et al. Sci Adv. 2019 Nov 27;5(11):eaax9115.

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