DR4004 | 5-HT7 antagonist | Probechem Biochemicals

Chemical Structure : DR4004

DR4004 (DR-4004)

Catalog No.: PC-22276Not For Human Use, Lab Use Only.

DR4004 (DR-4004) is a potent, highly selective 5-HT7 antagonist with bingding pKi of 8.67, >50-fold selectivity over the 5-HT2 receptor, and other 5-HT receptors.

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Biological Activity

DR4004 (DR-4004) hydrochloride is a potent, highly selective 5-HT7 antagonist with bingding pKi of 8.67, >50-fold selectivity over the 5-HT2 receptor, and other 5-HT receptors.

Physicochemical Properties

M.Wt	386.54
Formula	C26H30N2O
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Benz[cd]indol-2(1H)-one, 2a-[4-(3,6-dihydro-4-phenyl-1(2H)-pyridinyl)butyl]-2a,3,4,5-tetrahydro-

References

1. Ehlen JC, et al. J Neurosci. 2001 Jul 15;21(14):5351-7.

2. Kogan HA, et al. Eur J Pharmacol. 2002 Aug 2;449(1-2):105-11.

3. Chika Kikuchi, et al. J. Med. Chem. 1999, 42, 4, 533–535.

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DR4004 (DR-4004)

Biological Activity

Physicochemical Properties

References

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