Chemical Structure : DR4004
Catalog No.: PC-22276Not For Human Use, Lab Use Only.
DR4004 (DR-4004) is a potent, highly selective 5-HT7 antagonist with bingding pKi of 8.67, >50-fold selectivity over the 5-HT2 receptor, and other 5-HT receptors.
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DR4004 (DR-4004) hydrochloride is a potent, highly selective 5-HT7 antagonist with bingding pKi of 8.67, >50-fold selectivity over the 5-HT2 receptor, and other 5-HT receptors.
M.Wt | 386.54 | |
Formula | C26H30N2O | |
Appearance | Solid | |
Storage |
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Solubility |
10 mM in DMSO |
1. Ehlen JC, et al. J Neurosci. 2001 Jul 15;21(14):5351-7.
2. Kogan HA, et al. Eur J Pharmacol. 2002 Aug 2;449(1-2):105-11.
3. Chika Kikuchi, et al. J. Med. Chem. 1999, 42, 4, 533–535.
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