DREADD agonist compound 21 | hM3Dq agonist

Chemical Structure : DREADD agonist compound 21

CAS No.: 56296-18-5

DREADD agonist compound 21 (DREADD agonist 21, hM3Dq agonist)

Catalog No.: PC-42096Not For Human Use, Lab Use Only.

DREADD agonist compound 21 (hM3Dq agonist) is a potent, selective human muscarinic acetylcholine M3 receptor (hM3Dq) full agonist with EC50 of 1.7 nM.

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10 mg	$148	In stock
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Biological Activity

DREADD agonist compound 21 (hM3Dq agonist) is a potent, selective human muscarinic acetylcholine M3 receptor (hM3Dq) full agonist with EC50 of 1.7 nM.
hM3Dq-agonist-21 displays 3.5-fold selective over H1, 40-fold selective over 5HT2A, 100-fold selective over 5HT2C, 165-fold selective over α1A, and inactive at native human M3 receptor (hM3).

Physicochemical Properties

M.Wt	278.3516
Formula	C17H18N4
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	DMSO: ≥ 78 mg/mL
Chemical Name/SMILES	5H-Dibenzo[b,e][1,4]diazepine, 11-(1-piperazinyl)-

References

1. Chen X, et al. ACS Chem Neurosci. 2015 Mar 18;6(3):476-84.

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DREADD agonist compound 21 (DREADD agonist 21, hM3Dq agonist)

Biological Activity

Physicochemical Properties

References

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