Chemical Structure : DS-1971a
CAS No.:
1450595-86-4
DS-1971a
(DS1971a)
Catalog No. : PC-72189Not For Human Use, Lab Use Only.
DS-1971a (DS1971a) is a highly potent, selective NaV1.7 inhibitor with IC50 of 22.8 nM (hNaV1.7) and 59.4 nM (mNaV1.7).
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-7218901
Biological Activity
DS-1971a (DS1971a) is a highly potent, selective NaV1.7 inhibitor with IC50 of 22.8 nM (hNaV1.7) and 59.4 nM (mNaV1.7).
Physicochemical Properties
M.Wt
465.928
Formula
C20H21ClFN5O3S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
5-chloro-2-fluoro-4-(((1S,2R)-2-(1-methyl-1H-pyrazol-5-yl)cyclohexyl)oxy)-N-(pyrimidin-4-yl)benzenesulfonamide
References
1. Shinozuka T, et al. J Med Chem.
2. Asano D, et al. Xenobiotica.
3. Asano D, et al. Drug Metab Dispos.
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