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You are here:Home-Chemical Inhibitors & Agonists-GPCR-Motilin Receptor-DS-3801b
DS-3801b

Chemical Structure : DS-3801b

CAS No.: 1369412-66-7

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DS-3801b (DS3801b)

Catalog No.: PC-73242Not For Human Use, Lab Use Only.

DS-3801b is a potent, selective, non-macrolide GPR38 (motilin receptor) agonist with EC50 of 5.3 and 1.3 nM for human and rabbit GPR38 respectively.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    DS-3801b is a potent, selective, non-macrolide GPR38 (motilin receptor) agonist with EC50 of 5.3 and 1.3 nM for human and rabbit GPR38 respectively.
    DS-3801b is 11-fold more potent (EC50=7.3 nM) intestinal contractile activity than GSK962040 (EC50=82.6 nM).
    DS-3801b promoted intestinal contractile activity in rabbit duodenum muscle tissue.

    Physicochemical Properties

    M.Wt 465.638
    Formula C28H39N3O3
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (1r,4S)-4-(3-(hydroxymethyl)phenoxy)-N-methyl-N-(3-methyl-4-(((S)-3-methylpiperazin-1-yl)methyl)phenyl)cyclohexane-1-carboxamide

    References

    1. Toda N, et al. Bioorg Med Chem Lett. 2022 Mar 1;59:128554.

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