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Chemical Structure : DS17701585
Catalog No.: PC-38649Not For Human Use, Lab Use Only.
DS17701585 is a novel potent, highly selective EP300/CBP histone acetyltransferase inhibitor with IC50 of 0.15 uM.
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DS17701585 is a novel potent, highly selective EP300/CBP histone acetyltransferase inhibitor with IC50 of 0.15 uM.
DS17701585 shows dose-dependent inhibition of SRY-box transcription factor 2 (SOX2) mRNA expression in a human lung squamous cell carcinoma cell line LK2-xenografted mouse model.
| M.Wt | 482.555 | |
| Formula | C24H26N4O5S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Ryutaro Kanada, et al. Bioorg Med Chem Lett. 2022 Jun 15;66:128726.
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