DS17701585 | EP300/CBP inhibitor | Probechem Biochemicals

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Chemical Structure : DS17701585

DS17701585 (DS 17701585)

Catalog No.: PC-38649Not For Human Use, Lab Use Only.

DS17701585 is a novel potent, highly selective EP300/CBP histone acetyltransferase inhibitor with IC50 of 0.15 uM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

DS17701585 is a novel potent, highly selective EP300/CBP histone acetyltransferase inhibitor with IC50 of 0.15 uM.
DS17701585 shows dose-dependent inhibition of SRY-box transcription factor 2 (SOX2) mRNA expression in a human lung squamous cell carcinoma cell line LK2-xenografted mouse model.

Physicochemical Properties

M.Wt	482.555
Formula	C24H26N4O5S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-N-(1H-indazol-4-yl)-3-(1-(4-methoxyphenyl)cyclopentane-1-carbonyl)thiazolidine-4-carboxamide 1,1-dioxide

References

1. Ryutaro Kanada, et al. Bioorg Med Chem Lett. 2022 Jun 15;66:128726.

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DS17701585 (DS 17701585)

Biological Activity

Physicochemical Properties

References

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