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Dual DRAK1 and DRAK2 inhibitor 1

Chemical Structure : Dual DRAK1 and DRAK2 inhibitor 1

CAS No.: 1629227-34-4

Dual DRAK1 and DRAK2 inhibitor 1 (DRAK2/1 inhibitor)

Catalog No.: PC-38221Not For Human Use, Lab Use Only.

Dual DRAK1 and DRAK2 inhibitor 1 is a potent, dual DRAK2/1 inhibitor Kd value of 9/5 nM, respectively.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    Dual DRAK1 and DRAK2 inhibitor 1 is a potent, dual DRAK2/1 inhibitor Kd value of 9/5 nM, respectively.
    Dual DRAK1 and DRAK2 inhibitor 1 also is a functional inhibitor of DRAK2/1 enzymatic activity with IC50 of 0.86 and 2.25 uM.
    Dual DRAK1 and DRAK2 inhibitor 1 is a chemical tool compound to study DRAK1 and DRAK2 biology.

    Physicochemical Properties

    M.Wt 396.505
    Formula C22H24N2O3S
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    N-(5-(3,4-dimethoxyphenyl)thieno[2,3-b]pyridin-3-yl)cyclohexanecarboxamide

    References

    1. Ling-Jie Gao, et al. J Med Chem. 2014 Sep 25;57(18):7624-43.

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