EP-2825 | MRGPRD agonist | Probechem Biochemicals

Chemical Structure : EP-2825

EP-2825 (EP2825)

Catalog No.: PC-23537Not For Human Use, Lab Use Only.

EP-2825 is a potent, selective Mas-related G protein-coupled receptor MRGPRD agonist with EC50 of 211.6 nM at Gq in BRET assay.

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Biological Activity

EP-2825 is a potent, selective Mas-related G protein-coupled receptor MRGPRD agonist with EC50 of 211.6 nM at Gq in BRET assay.
EP-2825 displays low off-target activity at SSTR4 and GPR97 in a panel of 300 GPCRs.
EP-2825 activates MRGPRD much more potently than β-alanine and GABA.

Physicochemical Properties

M.Wt	428.96
Formula	C23H29ClN4O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-((1-(2-(4-chlorophenyl)-2-methylpropanoyl)piperidin-4-yl)amino)-5,6,7,8-tetrahydroquinazolin-4(3H)-one

References

1. Wang C, et al. Cell Rep. 2024 Nov 23;43(12):114942.

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EP-2825 (EP2825)

Biological Activity

Physicochemical Properties

References

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