EP300 degrader MC-1

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Chemical Structure : EP300 degrader MC-1

Catalog No.: PC-22345Not For Human Use, Lab Use Only.

EP300 degrader MC-1 is a specific, bifunctional small molecule EP300 degrader, preferentially degrades EP300 in a proteasome-dependent manner, does not degrade CREBBP.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

EP300 degrader MC-1 is a specific, bifunctional small molecule EP300 degrader, preferentially degrades EP300 in a proteasome-dependent manner, does not degrade CREBBP.

Physicochemical Properties

M.Wt	1062.35
Formula	C59H71N11O6S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(2S,4R)-1-((R)-2-(8-(2-(4-(6-((R)-2-(((S)-2-(4-cyanophenyl)propyl)amino)-2-phenylacetamido)pyridin-3-yl)-1H-pyrazol-1-yl)acetamido)octanamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-((S)-1-(4-(4-methylisothiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide

References

1. Xuemin Chen, et al. bioRxiv [Preprint]. 2024 May 5:2024.05.03.592353.

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