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EP300 degrader MC-1

Chemical Structure : EP300 degrader MC-1

CAS No.:

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EP300 degrader MC-1

Catalog No.: PC-22345Not For Human Use, Lab Use Only.

EP300 degrader MC-1 is a specific, bifunctional small molecule EP300 degrader, preferentially degrades EP300 in a proteasome-dependent manner, does not degrade CREBBP.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    EP300 degrader MC-1 is a specific, bifunctional small molecule EP300 degrader, preferentially degrades EP300 in a proteasome-dependent manner, does not degrade CREBBP.

    Physicochemical Properties

    M.Wt 1062.35
    Formula C59H71N11O6S
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (2S,4R)-1-((R)-2-(8-(2-(4-(6-((R)-2-(((S)-2-(4-cyanophenyl)propyl)amino)-2-phenylacetamido)pyridin-3-yl)-1H-pyrazol-1-yl)acetamido)octanamido)-3,3-dimethylbutanoyl)-4-hydroxy-N-((S)-1-(4-(4-methylisothiazol-5-yl)phenyl)ethyl)pyrrolidine-2-carboxamide

    References

    1. Xuemin Chen, et al. bioRxiv [Preprint]. 2024 May 5:2024.05.03.592353.

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