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Chemical Structure : ER-851
Catalog No.: PC-72059Not For Human Use, Lab Use Only.
ER-001259851-000 is a potent, selective, orally active Axl inhibitor with IC50 of 5.2 nM in cell free assays, displays >35-fold selectivity against Mer (IC50=190 nM).
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ER-001259851-000 (ER-851) is a potent, selective, orally active Axl inhibitor with IC50 of 5.2 nM in cell free assays, displays >35-fold selectivity against Mer (IC50=190 nM).
ER-001259851-000 shows a promising pharmacokinetic profile in mice.
| M.Wt | 668.774 | |
| Formula | C36H41FN8O4 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Satoshi Inoue, et al. Bioorg Med Chem Lett. 2021 Sep 15;48:128247.
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