Eclitasertib (DNL758, SAR443122) | RIPK1 inhibitor

Chemical Structure : Eclitasertib

CAS No.: 2125450-76-0

Catalog No.: PC-72533Not For Human Use, Lab Use Only.

Eclitasertib (DNL-758, SAR-443122) is a potent, orally bioavailable, small-molecule RIPK1 inhibitor with IC50 of <1 uM.

Packing	Price	Stock
5 mg	$228	In stock
10 mg	$368	In stock
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Biological Activity

Eclitasertib (DNL-758, SAR-443122) is a potent, orally bioavailable, small-molecule RIPK1 inhibitor with IC50 of <1 uM.

M.Wt	378.39
Formula	C19H18N6O3
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(S)-5-benzyl-N-(5-methyl-4-oxo-2,3,4,5-tetrahydropyrido[3,2-b][1,4]oxazepin-3-yl)-4H-1,2,4-triazole-3-carboxamide

1. WO2017136727A2, Example 42.