Welcome to ProbeChem!Global Supplier of Chemical Probes, Inhibitors & Agonists.
    English |     Chinese

Product Inquiry: sales@probechem.com
Order/PO receiving: order@probechem.com

You are here:Home-Chemical Inhibitors & Agonists-GPCR-5-HT Receptor-Eletriptan
Eletriptan

Chemical Structure : Eletriptan

CAS No.: 143322-58-1

Add to Favorites

Eletriptan (UK116044, UK 116044)

Catalog No.: PC-61868Not For Human Use, Lab Use Only.

Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist with pKi of 8.0 and 8.9.

Packing Price Stock Quantity
25 mg Get quote
50 mg Get quote
100 mg Get quote
Get Quotation Now
* Please select Quantity before adding items.
 or Bulk Inquiry

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist with pKi of 8.0 and 8.9.
    Eletriptan (UK 116044) significantly increases occluded wedge pressure and mean pulmonary artery pressure in vivo, with no significant coronary artery constriction, and obstructive coronary artery disease.
    Eletriptan (UK 116044) displays antimigraine activity.

    Physicochemical Properties

    M.Wt 382.52
    Formula C22H26N2O2S
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20 °C 12 Months; 4°C 6 Months
    In Solvent
    -80 °C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole

    References

    1. Napier C, et al. Eur J Pharmacol. 1999 Mar 5;368(2-3):259-68.

    2. Gupta P, et al. Eur J Pharmacol. 1999 Feb 19;367(2-3):283-90.

    3. Muir DF, et al. Clin Pharmacol Ther. 1999 Jul;66(1):85-90.

    Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

    Contact Us sales@probechem.com

    Bulk Inquiry

    * Indicates a Required FieldYour information is safe with us.

    • *Product name:
    • *Applicant name:
    • *Email address:
    • *Organization name:
    • *Requested quantity:
    • *Country:
    • *Additional Information:

    Get Quote

    * Indicates a Required FieldYour information is safe with us.

    • *Product name:
    • *Applicant name:
    • *Email address:
    • *Organization name:
    • *Requested quantity:
    • *Country:
    • Additional Information: