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Chemical Structure : Eletriptan
Catalog No.: PC-61868Not For Human Use, Lab Use Only.
Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist with pKi of 8.0 and 8.9.
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Eletriptan (UK 116044) is a potent, selective, and orally active 5-HT1B/1D receptor agonist with pKi of 8.0 and 8.9.
Eletriptan (UK 116044) significantly increases occluded wedge pressure and mean pulmonary artery pressure in vivo, with no significant coronary artery constriction, and obstructive coronary artery disease.
Eletriptan (UK 116044) displays antimigraine activity.
| M.Wt | 382.52 | |
| Formula | C22H26N2O2S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Napier C, et al. Eur J Pharmacol. 1999 Mar 5;368(2-3):259-68.
2. Gupta P, et al. Eur J Pharmacol. 1999 Feb 19;367(2-3):283-90.
3. Muir DF, et al. Clin Pharmacol Ther. 1999 Jul;66(1):85-90.
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