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Chemical Structure : Eletriptan hydrobromide
CAS No.: 177834-92-3
Catalog No.: PC-61867Not For Human Use, Lab Use Only.
Eletriptan (UK 116044) hydrobromide is a potent, selective, and orally active 5-HT1B/1D receptor agonist with Ki of 0.92 nM and 3.14 nM respectively.
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Eletriptan (UK 116044) hydrobromide is a potent, selective, and orally active 5-HT1B/1D receptor agonist with Ki of 0.92 nM and 3.14 nM respectively.
Eletriptan (UK 116044) significantly increases occluded wedge pressure and mean pulmonary artery pressure in vivo, with no significant coronary artery constriction, and obstructive coronary artery disease.
Eletriptan (UK 116044) displays antimigraine activity.
| M.Wt | 463.43 | |
| Formula | C22H26N2O2S.HBr | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
3-[[(2R)-1-Methyl-2-pyrrolidinyl]methyl]-5-[2-(phenylsulfonyl)ethyl]-1H-indole hydrobromide |
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1. Napier C, et al. Eur J Pharmacol. 1999 Mar 5;368(2-3):259-68.
2. Gupta P, et al. Eur J Pharmacol. 1999 Feb 19;367(2-3):283-90.
3. Muir DF, et al. Clin Pharmacol Ther. 1999 Jul;66(1):85-90.
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