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Emraclidine

Chemical Structure : Emraclidine

CAS No.: 2170722-84-4

Emraclidine (CVL-231, PF-06852231)

Catalog No.: PC-38388Not For Human Use, Lab Use Only.

Emraclidine (CVL-231) is a potent, selective positive allosteric modulator (PAM) of M4 muscarinic receptor subtype in development for schizophrenia.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

Emraclidine (CVL-231, PF-06852231) is a potent, selective positive allosteric modulator (PAM) of M4 muscarinic receptor subtype in development for schizophrenia.

Physicochemical Properties

M.Wt 390.410
Formula C20H21F3N4O
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

1-(2,4-dimethyl-5,7-dihydro-6H-pyrrolo[3,4-b]pyridin-6-yl)-2-(1-(2-(trifluoromethyl)pyridin-4-yl)azetidin-3-yl)ethan-1-one

References

1. Patent WO2018002760.

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