Eplerenone | Aldosterone receptor antagonist, MR antagonist

Chemical Structure : Eplerenone

CAS No.: 107724-20-9

Eplerenone (Epoxymexrenone)

Catalog No.: PC-27029Not For Human Use, Lab Use Only.

Eplerenone (Epoxymexrenone) is a selective, orally active aldosterone receptor antagonist, also is a selective mineralocorticoid receptor antagonist with IC50 of 81 nM.

Packing	Price	Stock
50 mg	$78	In stock
100 mg	$118	In stock
250 mg	$188	In stock
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Biological Activity

Eplerenone (Epoxymexrenone) is a selective, orally active aldosterone receptor antagonist, also is a selective mineralocorticoid receptor antagonist with IC50 of 81 nM.

Physicochemical Properties

M.Wt	414.50
Formula	C24H30O6
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	Methyl (4aS,4bR,5aR,6aS,7R,9aS,9bR,10R)-4a,6a-dimethyl-2,4'-dioxo-2,4,4a,4',5a,5',6,6a,8,9,9a,9b,10,11-tetradecahydro-3H,3'H-spiro[cyclopenta[1,2]phenanthro[4,4a-b]oxirene-7,2'-furan]-10-carboxylate

References

1. McMahon EG. Curr Opin Pharmacol. 2001 Apr;1(2):190-6.

2. Delyani JA, et al. Cardiovasc Drug Rev. 2001 Fall;19(3):185-200.

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Eplerenone (Epoxymexrenone)

Biological Activity

Physicochemical Properties

References

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