Etamicastat hydrochloride | Dopamine beta-hydroxylase inhibitor

Chemical Structure : Etamicastat hydrochloride

CAS No.: 677773-32-9

Etamicastat hydrochloride (BIA 5-453)

Catalog No.: PC-22597Not For Human Use, Lab Use Only.

Etamicastat hydrochloride (BIA 5-453 hydrochloride) is a potent, peripherally selective and reversible dopamine-β-hydroxylase (DβH) inhibitor with IC50 of 107 nM, reduces the biosynthesis of norepinephrine (noradrenaline).

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Biological Activity

Physicochemical Properties

M.Wt	347.81
Formula	C14H16ClF2N3OS
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-5-(2-aminoethyl)-1-(6,8-difluorochroman-3-yl)-1,3-dihydro-2H-imidazole-2-thione hydrochloride

References

1. Beliaev A, et al. J Med Chem. 2006 Feb 9;49(3):1191-7.

2. Loureiro AI, et al. Eur J Pharmacol. 2014 Oct 5;740:285-94.

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Etamicastat hydrochloride (BIA 5-453)

Biological Activity

Physicochemical Properties

References

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