Chemical Structure : Fosaprepitant dimeglumine
CAS No.: 265121-04-8
Catalog No.: PC-25517Not For Human Use, Lab Use Only.
Fosaprepitant dimeglumine (MK-0517) is a prodrug of Aprepitant (PC-42185), which is a potent, selective neurokinin-1 receptor (NK1R)antagonist
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| 50 mg | $148 | In stock | |
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Fosaprepitant dimeglumine (MK-0517) is a prodrug of Aprepitant (PC-42185), which is a potent, selective neurokinin-1 receptor (NK1R)antagonist
| M.Wt | 1004.84 | |
| Formula | C37H56F7N6O16P | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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| Chemical Name/SMILES |
(2R,3R,4R,5S)-6-(Methylamino)hexane-1,2,3,4,5-pentaol ((3-(((2R,3S)-2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-3-(4-fluorophenyl)morpholino)methyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)phosphonate)(2:1) |
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1. Bayati S, et al. Eur J Pharmacol. 2016 Nov 15;791:274-283.
2. Pranav Prasoon, et al. Indian J Pharmacol. 2016 Jul-Aug; 48(4): 394-398.
3. Navari RM. Expert Opin Investig Drugs. 2007 Dec;16(12):1977-85.

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