Catalog No.: PC-42736Not For Human Use, Lab Use Only.
Danegaptide (GAP-134, ZP1609) is a potent, orally active gap-junction modifier, prevents significantly conduction velocity slowing at 10 nM compared with vehicle.
Danegaptide (GAP-134, ZP1609) is a potent, orally active gap-junction modifier, prevents significantly conduction velocity slowing at 10 nM compared with vehicle.
Danegaptide (GAP-134, ZP1609) has highly desirable in vitro and in vivo safety profile including (1) lack of direct effects on membrane ion currents, hERG inhibition, and CYP450 liabilities, (2) negative AMES result, (3) a benign NovaScreen profile, and (4) no effects on systemic hemodynamics.
