GD136 (VUF10775) | H1R/H4R antagonist | Probechem Biochemicals

Chemical Structure : GD136

GD136 (GD-136, VUF10775, VUF-10775)

Catalog No.: PC-28138Not For Human Use, Lab Use Only.

GD136 (GD-136) is a potent, selective dual histamine H1 and H4 receptors (H1R/H4R) ligand / antagonist with pKi of 7.61 and 7.93 (hH1R/hH4R), shows >100-fold selectivity over hH2R and hH3R.

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Biological Activity

GD136 (VUF10775, GD-136) is a potent, selective dual histamine H1 and H4 receptors (H1R/H4R) ligand / antagonist with pKi of 7.61 and 7.93 (hH1R/hH4R), shows >100-fold selectivity over hH2R and hH3R.

Physicochemical Properties

M.Wt	494.54
Formula	C22H25F3N6O2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	2-((2-(4-methylpiperazin-1-yl)-5-(trifluoromethyl)quinazolin-4-yl)amino)-N-phenylethane-1-sulfonamide

References

1. Weber P, et al. J Med Chem. 2026 Sep 10;69(17):20967-21003.

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GD136 (GD-136, VUF10775, VUF-10775)

Biological Activity

Physicochemical Properties

References

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