GD136 hydrochloride | H1R/H4R antagonist

Chemical Structure : GD136 hydrochloride

GD136 hydrochloride (VUF10775, GD-136)

Catalog No.: PC-28139Not For Human Use, Lab Use Only.

GD136 hydrochloride (VUF10775, GD-136) is a potent, selective dual histamine H1 and H4 receptors (H1R/H4R) ligand / antagonist with pKi of 7.61 and 7.93 (hH1R/hH4R), shows >100-fold selectivity over hH2R and hH3R.

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Biological Activity

Physicochemical Properties

M.Wt	531.00
Formula	C22H26ClF3N6O2S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	2-((2-(4-Methylpiperazin-1-yl)-5-(trifluoromethyl)quinazolin-4-yl)amino)-N-phenylethane-1-sulfonamide hydrochloride

References

1. Weber P, et al. J Med Chem. 2026 Sep 10;69(17):20967-21003.

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GD136 hydrochloride (VUF10775, GD-136)

Biological Activity

Physicochemical Properties

References

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