GEn-1124 | p38α/MK2 modulator | Probechem Biochemicals

Chemical Structure : GEn-1124

GEn-1124 (GEn1124, SF-7-044 dihydrochloride dihydrate)

Catalog No.: PC-23072Not For Human Use, Lab Use Only.

GEn-1124 is a first-in-class small molecule modulator of p38α/MK2 signaling targeted to a pocket near the ED substrate binding domain of p38α, destabilizes the MK2: p38 complex.

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Biological Activity

GEn-1124 is a first-in-class small molecule modulator of p38α/MK2 signaling targeted to a pocket near the ED substrate binding domain of p38α, destabilizes the MK2: p38 complex.

Physicochemical Properties

M.Wt	534.49
Formula	C23H33Cl2N3O5S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	5-(dimethylamino)-N-(4-(morpholinomethyl)phenyl)naphthalene-1-sulfonamide dihydrochloride dihydrate

References

1. Tulapurkar ME, et al. J Pharmacol Exp Ther. 2024 Sep 16:JPET-AR-2024-002281.

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GEn-1124 (GEn1124, SF-7-044 dihydrochloride dihydrate)

Biological Activity

Physicochemical Properties

References

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