Chemical Structure : GLPG0187
CAS No.:
1320346-97-1
GLPG0187
(GLPG 0187, GLPG-0187)
Catalog No. : PC-42179Not For Human Use, Lab Use Only.
GLPG0187 (GLPG 0187) is a highly potent, broad spectrum integrin receptor antagonist with IC50 of 1-10 nM for αvβ1, αvβ3, αvβ5, αvβ6, αvβ8 and α5β1.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4217901
Biological Activity
GLPG0187 (GLPG 0187) is a highly potent, broad spectrum integrin receptor antagonist with IC50 of 1-10 nM for αvβ1, αvβ3, αvβ5, αvβ6, αvβ8 and α5β1.
Physicochemical Properties
M.Wt
595.713
Formula
C29H37N7O5S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: 15 mg/mL
Chemical Name/SMILES
L-Alanine, 3-[[2,5-dimethyl-6-[4-(5,6,7,8-tetrahydro-1,8-naphthyridin-2-yl)-1-piperidinyl]-4-pyrimidinyl]amino]-N-[(4-methoxyphenyl)sulfonyl]-
References
1. Pujuguet P, et al. Eur J Cancer.
2. Cirkel GA, et al. Invest New Drugs.
3. van der Horst G, et al. Neoplasia.
4. Reeves KJ, et al. Int J Cancer.
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