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GLPG0492

Chemical Structure : GLPG0492

CAS No.: 1215085-92-9

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GLPG0492 (GLPG-0492)

Catalog No.: PC-45421Not For Human Use, Lab Use Only.

GLPG0492 is an orally active, non-steroidal selective androgen receptor modulator (SARM) with in vitro potency of 13 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

GLPG0492 is an orally active, non-steroidal selective androgen receptor modulator (SARM) with in vitro potency of 13 nM.
GLPG0492 exhibits anabolic activity on muscle, strongly dissociated from the androgenic activity on prostate in a classical model of orchidectomized rat.
GLPG0492 shows a potential treatment for Duchenne muscular dystrophy (DMD).

Physicochemical Properties

M.Wt 389.328
Formula C19H14F3N3O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

Benzonitrile, 4-[(4S)-4-(hydroxymethyl)-3-methyl-2,5-dioxo-4-phenyl-1-imidazolidinyl]-2-(trifluoromethyl)-

References

1. Nique F, et al. J Med Chem. 2012 Oct 11;55(19):8236-47.

2. Cozzoli A, et al. Pharmacol Res. 2013 Jun;72:9-24.

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