Chemical Structure : GLPG0974
CAS No.:
1391076-61-1
GLPG0974
(GLPG-0974)
Catalog No. : PC-62591Not For Human Use, Lab Use Only.
GLPG 0974 is a potent, selective free fatty acid receptor 2 (FFA2, GPR43) antagonist with IC50 of 95 nM.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-6259101
Biological Activity
GLPG0974 is a potent, selective free fatty acid receptor 2 (FFA2, GPR43 ) antagonist with IC50 of 95 nM.
Physicochemical Properties
M.Wt
484.995
Formula
C25H25ClN2O4S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
4-[[[(2R)-1-(Benzo[b]thien-3-ylcarbonyl)-2-methyl-2-azetidinyl]carbonyl][(3-chlorophenyl)
References
1. Pizzonero M, et al. J Med Chem.
2. Sergeev E, et al. J Biol Chem.
3. Namour F, et al. Br J Clin Pharmacol.
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