You are here:Home-Chemical Inhibitors & Agonists-GPCR-GPR183 (EBI2)-GPR183 antagonist SAE-1
GPR183 antagonist SAE-1

Chemical Structure : GPR183 antagonist SAE-1

CAS No.: 1210803-60-3

GPR183 antagonist SAE-1 (SAE-1)

Catalog No.: PC-72118Not For Human Use, Lab Use Only.

GPR183 antagonist SAE-14 is a potent, selective GPR183 antagonist with IC50 of 8.3 nM, inhibits calcium mobilization induced by 7α,25-OHC in HL-60 cells.

Packing Price Stock Quantity
25 mg Get quote
50 mg Get quote
100 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    GPR183 antagonist SAE-14 is a potent, selective GPR183 antagonist with IC50 of 8.3 nM, inhibits calcium mobilization induced by 7α,25-OHC in HL-60 cells.

    Physicochemical Properties

    M.Wt 375.425
    Formula C19H25N3O5
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-(1-(3,4,5-trimethoxyphenyl)ethyl)acetamide

    References

    1. Kathryn Braden, et al. J Pharmacol Exp Ther. 2020 Nov;375(2):367-375.

    Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

    Contact Us sales@probechem.com

    Bulk Inquiry

    * Indicates a Required FieldYour information is safe with us.

    • *Product name:
    • *Applicant name:
    • *Email address:
    • *Organization name:
    • *Requested quantity:
    • *Country:
    • *Additional Information:

    Get Quote

    * Indicates a Required FieldYour information is safe with us.

    • *Product name:
    • *Applicant name:
    • *Email address:
    • *Organization name:
    • *Requested quantity:
    • *Country:
    • Additional Information: