GPR183 inverse agonist compound 78 | GPR183 inverse agonist

Chemical Structure : GPR183 inverse agonist compound 78

GPR183 inverse agonist compound 78 (GPR183 inverse agonist 1)

Catalog No.: PC-27089Not For Human Use, Lab Use Only.

GPR183 inverse agonist 1 (Compound 78) is a seletive GPR183 inverse agonist, inhibits the GPR183-mediated Gi activation with pIC50 of 6.29, modulates both Gi and β-arrestin2-responses of GPR183.

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Biological Activity

GPR183 inverse agonist 1 (Compound 78) is a seletive GPR183 inverse agonist, inhibits the GPR183-mediated Gi activation with pIC50 of 6.29, modulates both Gi and β-arrestin2-responses of GPR183.

Physicochemical Properties

M.Wt	442.32
Formula	C20H20BrN5O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	2-((1-(4-bromobenzoyl)piperidin-4-yl)methyl)-6-(1H-pyrazol-1-yl)pyridazin-3(2H)-one

References

1. Andersson L, et al. Nat Commun. 2026 May 30. doi: 10.1038/s41467-026-73857-9.

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