GPR40 agonist AP4

Chemical Structure : GPR40 agonist AP4

Catalog No.: PC-20869Not For Human Use, Lab Use Only.

GPR40 agonist AP4 is a potent, selective, full allosteric agonist (AgoPAM) of GPR40 with EC50 of 0.08 nM, Emax=283%.

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Purity & Documentation Purity: >98% (HPLC)

Biological Activity

GPR40 agonist AP4 is a potent, selective, full allosteric agonist (AgoPAM) of GPR40 with EC50 of 0.08 nM, Emax=283%.

M.Wt	574.74
Formula	C35H43FN2O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	O=C(O)[C@@H](C)[C@@H](C1CC1)C2=CC3=C(C=C2)CC[C@H](C4=CC=C(C5=CC(OC)=NC=C5F)C(CN(C(C)C)C(C)C)=C4)O3

1. Jun Lu, et al. GPR40 agonist AP8, Nat Struct Mol Biol . 2017 Jul;24(7):570-577.

2. Patent WO2016022742 A1.