GPR55 agonist 28

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Chemical Structure : GPR55 agonist 28

Catalog No.: PC-21153Not For Human Use, Lab Use Only.

GPR55 agonist 28 is a potent, selective GPR55 agonist with EC50 of 131 and 141 nM for human and rat GPR55, respectively, in Ca2+ flux assays.

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Biological Activity

GPR55 agonist 28 is a potent, selective GPR55 agonist with EC50 of 131 and 141 nM for human and rat GPR55, respectively, in Ca2+ flux assays.
GPR55 agonist 28 activates the β-arrestin pathway with EC50 of 6.2 nM, produces a full activation of hGPR55 in the Ca2+ flux assay (Emax: 105%).
GPR55 agonist 28 (10 uM) markedly decreased the frequency of rat MSN cell firing in cultured rodent striatal MSNs.

Physicochemical Properties

M.Wt	365.37
Formula	C19H16FN5O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-5-(3-((1-(4-Fluorophenyl)ethyl)amino)-1,2,4-triazin-6-yl)-3-methylbenzo[d]oxazol-2(3H)-one

References

1. Richard C. Hewer, et al. J. Med. Chem. 2023.

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GPR55 agonist 28

Biological Activity

Physicochemical Properties

References

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