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Chemical Structure : GPR55 agonist 28
Catalog No.: PC-21153Not For Human Use, Lab Use Only.
GPR55 agonist 28 is a potent, selective GPR55 agonist with EC50 of 131 and 141 nM for human and rat GPR55, respectively, in Ca2+ flux assays.
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GPR55 agonist 28 is a potent, selective GPR55 agonist with EC50 of 131 and 141 nM for human and rat GPR55, respectively, in Ca2+ flux assays.
GPR55 agonist 28 activates the β-arrestin pathway with EC50 of 6.2 nM, produces a full activation of hGPR55 in the Ca2+ flux assay (Emax: 105%).
GPR55 agonist 28 (10 uM) markedly decreased the frequency of rat MSN cell firing in cultured rodent striatal MSNs.
| M.Wt | 365.37 | |
| Formula | C19H16FN5O2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Richard C. Hewer, et al. J. Med. Chem. 2023.
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