Chemical Structure : GR127935 hydrochloride
CAS No.:
148642-42-6
GR127935 hydrochloride
(GR-127935 hydrochloride)
Catalog No. : PC-61866Not For Human Use, Lab Use Only.
GR-127935 potent and selective 5-HT1B/1D receptor antagonist with pKi of 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptor.
Packing Price Stock Quantity 5 mg $98 In stock 0 1 2 3 4 5 10 mg $148 In stock 0 1 2 3 4 5 25 mg $258 In stock 0 1 2 3 4 5 50 mg Get quote 0 1 2 3 4 5 100 mg Get quote 0 1 2 3 4 5
Bulk size, bulk discount!
Welcome credit card payment!
E-mail: sales@probechem.com
Tech Support: tech@probechem.com
Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-6186601
Biological Activity
GR127935 hydrochloride is a potent and selective 5-HT1B/1D receptor antagonist with pKi of 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptor.
Physicochemical Properties
M.Wt
534.06
Formula
C29H31N5O3.HCl
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
N-[4-methoxy-3-(4-methylpiperazin-1-yl)phenyl]-4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]benzamide hydrochloride
References
1. Clitherow JW, et al. J Med Chem
2. Knobelman DA, et al. J Pharmacol Exp Ther.
3. De Vries P, et al. Br J Pharmacol.
Contact Us
sales@probechem.com
