GSK-1440115 | Urotensin II receptor antagonist

Chemical Structure : GSK-1440115

GSK-1440115 (GSK1440115)

Catalog No.: PC-28271Not For Human Use, Lab Use Only.

GSK-1440115 is a potent, nonpeptidic antagonist of Urotensin II receptor (UT) with pKi of 7.34-8.64 across species, shows competitive antagonism at UT in arteries with pA2 of 5.59-7.71.

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Biological Activity

GSK-1440115 is a potent, nonpeptidic antagonist of Urotensin II receptor (UT) with pKi of 7.34-8.64 across species, shows competitive antagonism at UT in arteries with pA2 of 5.59-7.71.

Physicochemical Properties

M.Wt	598.48
Formula	C30H29Cl2N3O6
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-4'-(1-(2-(6,7-dichloro-3-oxo-2,3-dihydro-4H-benzo[b][1,4]oxazin-4-yl)-N-methylacetamido)-2-morpholinoethyl)-[1,1'-biphenyl]-4-carboxylic acid

References

1. Behm DJ, et al. Br J Pharmacol. 2010 Sep;161(1):207-28.

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GSK-1440115 (GSK1440115)

Biological Activity

Physicochemical Properties

References

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