GSK1034702 |CAS:932373-87-0 Probechem Biochemicals

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Chemical Structure : GSK1034702

CAS No.: 932373-87-0

GSK1034702 (GSK-1034702;GSK 1034702)

Catalog No.: PC-35626Not For Human Use, Lab Use Only.

GSK1034702 (GSK-1034702) is a potent, allosteric M1 receptor agonist, inhibits binding of [3H]-NMS (0.5 nM) to M1 mAChR with pKi of 6.5.

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10 mg	$328	In stock
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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

GSK1034702 (GSK-1034702) is a potent, allosteric M1 receptor agonist, inhibits binding of [3H]-NMS (0.5 nM) to M1 mAChR with pKi of 6.5.
GSK1034702 improves memory encoding potentially by modulating hippocampal function.

Physicochemical Properties

M.Wt	333.407
Formula	C18H24FN3O2
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	7-fluoro-5-methyl-3-[1-(oxan-4-yl)piperidin-4-yl]-1H-benzimidazol-2-one

References

1. Nathan PJ, et al. Int J Neuropsychopharmacol. 2013 May;16(4):721-31.

2. Bradley SJ, et al. Mol Pharmacol. 2018 Jun;93(6):645-656.

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GSK1034702 (GSK-1034702;GSK 1034702)

Biological Activity

Physicochemical Properties

References

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