You are here:Home-Chemical Inhibitors & Agonists-Metabolic Enzyme/Protease-Protein Arginine Deiminase (PAD)-GSK121 trifluoroacetate
GSK121 trifluoroacetate

Chemical Structure : GSK121 trifluoroacetate

CAS No.: 1652591-80-4

GSK121 trifluoroacetate (GSK121 TFA)

Catalog No.: PC-38517Not For Human Use, Lab Use Only.

GSK121 TFA salt is a small molecule inhibitor of potein arginine deiminase 4 (PAD4) with IC50 of 3.2 uM.

Packing Price Stock Quantity
5 mg $148 In stock
10 mg $228 In stock
25 mg $388 In stock
50 mg Get quote
100 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

GSK121 TFA salt is a small molecule inhibitor of potein arginine deiminase 4 (PAD4) with IC50 of 3.2 uM.

Physicochemical Properties

M.Wt 501.510
Formula C25H26F3N5O3
Appearance Solid
CAS No.
Storage
Solide Powder
-20°C 12 Months; 4°C 6 Months
In Solvent
-80°C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO

Chemical Name/SMILES

(3-aminopiperidin-1-yl)(1-methyl-2-(1-methyl-1H-indol-2-yl)-1H-benzo[d]imidazol-5-yl)methanone 2,2,2-trifluoroacetate

References

1. Drewes G, et al. Nat Chem Biol. 2015 Mar;11(3):189-91.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: