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Chemical Structure : GSK1292263
CAS No.: 1032823-75-8
Catalog No.: PC-42879Not For Human Use, Lab Use Only.
GSK1292263 is a novel potent, selective GPR119 agonist with pEC50 of 6.9 and 6.7 for human and rat GPR119, respectively.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $98 | In stock | |
| 25 mg | $158 | In stock | |
| 50 mg | $258 | In stock | |
| 100 mg | Get quote |
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GSK1292263 is a novel potent, selective GPR119 agonist with pEC50 of 6.9 and 6.7 for human and rat GPR119, respectively.
GSK1292263 elevates circulating glucose-dependent insulinotropic peptide, GLP-1 and peptide tyrosine-tyrosine in nonclinical models of diabetes, with no effect on plasma glucose.
| M.Wt | 456.5578 | |
| Formula | C23H28N4O4S | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: ≥ 30 mg/mL |
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| Chemical Name/SMILES |
Pyridine, 5-[[1-[3-(1-methylethyl)-1,2,4-oxadiazol-5-yl]-4-piperidinyl]methoxy]-2-[4-(methylsulfonyl)phenyl]- |
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1. Polli JW, et al. Xenobiotica. 2013 Jun;43(6):498-508.
2. Nunez DJ, et al. PLoS One. 2014 Apr 3;9(4):e92494.
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