Chemical Structure : GSK1904529A
CAS No.:
1089283-49-7
GSK1904529A
(GSK-1904529A, GSK 1904529A)
Catalog No. : PC-42636Not For Human Use, Lab Use Only.
GSK1904529A is a potent, selective, ATP-competitive inhibitor of IGF-1R and IR with IC50 of 27 nM and 25 nM.
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4263601
Biological Activity
GSK1904529A is a potent, selective, ATP-competitive inhibitor of IGF-1R and IR with IC50 of 27 nM and 25 nM.
Physicochemical Properties
M.Wt
851.9631
Formula
C44H47F2N9O5S
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
10 mM in DMSO
Chemical Name/SMILES
Benzamide, N-(2,6-difluorophenyl)-5-[3-[2-[[5-ethyl-2-methoxy-4-[4-[4-(methylsulfonyl)-1-piperazinyl]-1-piperidinyl]phenyl]amino]-4-pyrimidinyl]imidazo[1,2-a]pyridin-2-yl]-2-methoxy-
References
1. Sabbatini P, et al. Clin Cancer Res.
2. Zhou Q, et al. Mol Med Rep.
3. Fei HD, et al. Oncotarget.
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