GSK251 | PI3Kδ inhibitor | Probechem Biochemicals

Chemical Structure : GSK251

CAS No.: 2125968-05-8

Catalog No.: PC-72781Not For Human Use, Lab Use Only.

GSK251 is a highly potent, selective, orally bioavailable inhibitor of PI3Kδ with pKi of 10.9, >1,000-fold selectivity over other PI3K isoforms.

Packing	Price	Stock
2 mg	$278	In stock
5 mg	$498	In stock
10 mg	$788	In stock
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Biological Activity

GSK251 is a highly potent, selective, orally bioavailable inhibitor of PI3Kδ with pKi of 10.9, >1,000-fold selectivity over other PI3K isoforms.

M.Wt	584.711
Formula	C29H37FN6O4S
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(2-(2-fluoro-4-((4-isopropylpiperazin-1-yl)methyl)phenyl)pyridin-4-yl)-2-methoxy-5-morpholinopyridine-3-sulfonamide

1. Kenneth Down, et al. J. Med. Chem. 2021, 64, 18, 13780–13792.