Chemical Structure : GSK2606414
CAS No.:
1337531-36-8
GSK2606414
(GSK 2606414, GSK-2606414)
Catalog No. : PC-45410Not For Human Use, Lab Use Only.
GSK2606414 is an orally available, potent, and selective PERK inhibitor with IC50 of 0.4 nM.
Packing Price Stock Quantity 5 mg $98 In stock 0 1 2 3 4 5 10 mg $148 In stock 0 1 2 3 4 5 25 mg $258 In stock 0 1 2 3 4 5 50 mg $428 In stock 0 1 2 3 4 5 100 mg Get quote 0 1 2 3 4 5
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Purity & Documentation Purity:
>98% (HPLC) Select Batch: PC-4541001
Biological Activity
GSK2606414 is an orally available, potent, and selective PERK inhibitor with IC50 of 0.4 nM.
Physicochemical Properties
M.Wt
451.4437
Formula
C24H20F3N5O
Appearance
Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility
DMSO: ≥ 31 mg/mL
Chemical Name/SMILES
Ethanone, 1-[5-(4-amino-7-methyl-7H-pyrrolo[2,3-d]pyrimidin-5-yl)-2,3-dihydro-1H-indol-1-yl]-2-[3-(trifluoromethyl)phenyl]-
References
1. Axten JM, et al. J Med Chem.
2. Ounallah-Saad H, et al. J Neurosci.
3. Guthrie LN, et al. J Biol Chem.
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