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GSK2881078

Chemical Structure : GSK2881078

CAS No.: 1539314-06-1

GSK2881078 (GSK-2881078, GSK 2881078)

Catalog No.: PC-42075Not For Human Use, Lab Use Only.

GSK2881078 potent and selective androgen receptor modulator (SARM), act as partial AR agonist and induces AR-mediated transcriptional activation in PC3(AR)2 cells with EC50 of 3.99 nM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

GSK2881078 is a potent and selective androgen receptor modulator (SARM), act as partial AR agonist and induces AR-mediated transcriptional activation in PC3(AR)2 cells with EC50 of 3.99 nM.

Physicochemical Properties

M.Wt 330.3254
Formula C14H13F3N2O2S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

DMSO: ≥ 33 mg/mL

Chemical Name/SMILES

1H-Indole-5-carbonitrile, 1-[(1R)-1-methyl-2-(methylsulfonyl)ethyl]-4-(trifluoromethyl)-

References

1. Neil D, et al. J Clin Endocrinol Metab. 2018;103(9):3215-3224.

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