You are here:Home-Chemical Inhibitors & Agonists-Nuclear Receptor/Transcription Factor-Androgen Receptor (AR)-GSK2881078
GSK2881078

Chemical Structure : GSK2881078

CAS No.: 1539314-06-1

GSK2881078 (GSK-2881078, GSK 2881078)

Catalog No.: PC-42075Not For Human Use, Lab Use Only.

GSK2881078 potent and selective androgen receptor modulator (SARM), act as partial AR agonist and induces AR-mediated transcriptional activation in PC3(AR)2 cells with EC50 of 3.99 nM.

Packing Price Stock Quantity
10 mg $128 In stock
25 mg $218 In stock
50 mg Get quote
100 mg Get quote

Bulk size, bulk discount!

E-mail: sales@probechem.com

Tech Support: tech@probechem.com

Purity & Documentation Purity: >98% (HPLC) Select Batch:

Biological Activity

GSK2881078 is a potent and selective androgen receptor modulator (SARM), act as partial AR agonist and induces AR-mediated transcriptional activation in PC3(AR)2 cells with EC50 of 3.99 nM.

Physicochemical Properties

M.Wt 330.3254
Formula C14H13F3N2O2S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

DMSO: ≥ 33 mg/mL

Chemical Name/SMILES

1H-Indole-5-carbonitrile, 1-[(1R)-1-methyl-2-(methylsulfonyl)ethyl]-4-(trifluoromethyl)-

References

1. Neil D, et al. J Clin Endocrinol Metab. 2018;103(9):3215-3224.

Copyright © 2022 probechem.com. All Rights Reserved. probechem Copyright

Contact Us sales@probechem.com

Bulk Inquiry

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • *Additional Information:

Get Quote

* Indicates a Required FieldYour information is safe with us.

  • *Product name:
  • *Applicant name:
  • *Email address:
  • *Organization name:
  • *Requested quantity:
  • *Country:
  • Additional Information: