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Chemical Structure : GSK962040
CAS No.: 923565-21-3
Catalog No.: PC-42738Not For Human Use, Lab Use Only.
GSK962040 (Camicinal) is a potent, selective, small molecule motilin receptor agonist with pEC50 of 7.9 (hMTL-R).
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 5 mg | $238 | In stock | |
| 10 mg | $388 | In stock | |
| 25 mg | $598 | In stock | |
| 50 mg | Get quote | ||
| 100 mg | Get quote |
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GSK962040 (Camicinal) is a potent, selective, small molecule motilin receptor (GPR38) agonist with pEC50 of 7.9 (hMTL-R).
GSK962040 displays selectivity over closely related human ghrelin acceptor (pEC50< 6.0) and no liabilities at the hERG channel.
GSK962040 possesses highly excellent pharmacokinetic profiles in both rat and dog.
| M.Wt | 424.5541 | |
| Formula | C25H33FN4O | |
| Appearance | Solid | |
| Storage |
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| Solubility |
DMSO: 12.73 mg/mL (Need ultrasonic) |
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| Chemical Name/SMILES |
Ethanone, 1-[4-[(3-fluorophenyl)amino]-1-piperidinyl]-2-[4-[[(3S)-3-methyl-1-piperazinyl]methyl]phenyl]- |
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1. Westaway SM, et al. J Med Chem. 2009 Feb 26;52(4):1180-9.
2. Sanger GJ, et al. Neurogastroenterol Motil. 2009 Jun;21(6):657-64, e30-1.
3. Broad J, et al. Br J Pharmacol. 2012 Oct;167(4):763-74.
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