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GSTO1 inhibitor C1-27

Chemical Structure : GSTO1 inhibitor C1-27

CAS No.: 568544-03-6

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GSTO1 inhibitor C1-27

Catalog No.: PC-61194Not For Human Use, Lab Use Only.

GSTO1 inhibitor C1-27 is a potent, selective, covalent glutathione S-transferase omega 1 (GSTO1) inhibitor with IC50 of 31 nM.

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Biological Activity

GSTO1 inhibitor C1-27 is a potent, selective, covalent glutathione S-transferase omega 1 (GSTO1) inhibitor with IC50 of 31 nM.
GSTO1 inhibitor C1-27 displays selective inhibition of the GSTO1 against several other cysteine-containing proteins at 1 uM.
GSTO1 inhibitor C1-27 suppresses cancer cell growth, enhances the cytotoxic effects of cisplatin and inhibits tumour growth in colon cancer models as single agent.

Physicochemical Properties

M.Wt 311.177
Formula C10H12Cl2N2O3S
Appearance Solid
CAS No.
Storage
Solide Powder
-20 °C 12 Months; 4°C 6 Months
In Solvent
-80 °C 6 Months; -20°C 6 Months
Shipping
Solubility

10 mM in DMSO
Chemical Name/SMILES

2-chloro-N-(4-chloro-3-(N,N-dimethylsulfamoyl)phenyl)acetamide

References

1. Ramkumar K, et al. Nat Commun. 2016 Oct 5;7:13084.

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