GW-5823 | CCK1 agonist | Probechem Biochemicals

Chemical Structure : GW-5823

GW-5823 (GW5823)

Catalog No.: PC-22019Not For Human Use, Lab Use Only.

GW5823 (GW-5823) a potent, selective orally active, gut-selective CCK1 receptor (CCK-A receptor) agonist with binding pIC50 of 7.64, ED50 of 109 nM in functional assays.

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Biological Activity

GW5823 (GW-5823) a potent, selective orally active, gut-selective CCK1 receptor (CCK-A receptor) agonist with binding pIC50 of 7.64, ED50 of 109 nM in functional assays.
GW5823 displays 50-fold selectivity over CCK-B receptor.

Physicochemical Properties

M.Wt	587.68
Formula	C35H33N5O4
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
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Solubility	10 mM in DMSO
Chemical Name/SMILES	2-(3-((2H-indazol-3-yl)methyl)-2,4-dioxo-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[b][1,4]diazepin-1-yl)-N-isopropyl-N-(4-methoxyphenyl)acetamide

References

1. Richard L Elliott, et al. Bioorg Med Chem Lett. 2010 Nov 15;20(22):6797-801.

2. B R Henke, et al. J Med Chem. 1997 Aug 15;40(17):2706-25.

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GW-5823 (GW5823)

Biological Activity

Physicochemical Properties

References

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