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GZ-794A

Chemical Structure : GZ-794A

CAS No.: 1392205-38-7

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GZ-794A (GZ794A)

Catalog No.: PC-47109Not For Human Use, Lab Use Only.

GZ-794A is a potent, selective inhibitor of vesicular monoamine transporter-2 (VMAT2) with Ki of 30 nM, inhibits methamphetamine-evoked endogenous dopamine release with IC50 of 0.4 uM.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    GZ-794A is a potent, selective inhibitor of vesicular monoamine transporter-2 (VMAT2) with Ki of 30 nM, inhibits methamphetamine-evoked endogenous dopamine release with IC50 of 0.4 uM.
    GZ-794A shows potential for treatment for methamphetamine abuse.

    Physicochemical Properties

    M.Wt 467.653
    Formula C32H37NO2
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO
    Chemical Name/SMILES

    (R)-3-[2,6-cis-di(1-naphthylethyl)piperidin-1-yl]propane-1,2-diol

    References

    1. Horton DB, et al. J Pharmacol Exp Ther. 2011 Oct;339(1):286-97.

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