GZ-794A | VMAT2 inhibitor | Probechem Biochemicals

Chemical Structure : GZ-794A

GZ-794A (GZ794A)

Catalog No.: PC-47109Not For Human Use, Lab Use Only.

GZ-794A is a potent, selective inhibitor of vesicular monoamine transporter-2 (VMAT2) with Ki of 30 nM, inhibits methamphetamine-evoked endogenous dopamine release with IC50 of 0.4 uM.

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Biological Activity

GZ-794A is a potent, selective inhibitor of vesicular monoamine transporter-2 (VMAT2) with Ki of 30 nM, inhibits methamphetamine-evoked endogenous dopamine release with IC50 of 0.4 uM.
GZ-794A shows potential for treatment for methamphetamine abuse.

Physicochemical Properties

M.Wt	467.653
Formula	C32H37NO2
Appearance	Solid
CAS No.
Storage	Solide Powder -20°C 12 Months; 4°C 6 Months	In Solvent -80°C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	(R)-3-[2,6-cis-di(1-naphthylethyl)piperidin-1-yl]propane-1,2-diol

References

1. Horton DB, et al. J Pharmacol Exp Ther. 2011 Oct;339(1):286-97.

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GZ-794A (GZ794A)

Biological Activity

Physicochemical Properties

References

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