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Chemical Structure : GZ-794A
Catalog No.: PC-47109Not For Human Use, Lab Use Only.
GZ-794A is a potent, selective inhibitor of vesicular monoamine transporter-2 (VMAT2) with Ki of 30 nM, inhibits methamphetamine-evoked endogenous dopamine release with IC50 of 0.4 uM.
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GZ-794A is a potent, selective inhibitor of vesicular monoamine transporter-2 (VMAT2) with Ki of 30 nM, inhibits methamphetamine-evoked endogenous dopamine release with IC50 of 0.4 uM.
GZ-794A shows potential for treatment for methamphetamine abuse.
| M.Wt | 467.653 | |
| Formula | C32H37NO2 | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
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1. Horton DB, et al. J Pharmacol Exp Ther. 2011 Oct;339(1):286-97.
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