GeA-69 | PARP14 inhibitor | Probechem Biochemicals

Chemical Structure : GeA-69

CAS No.: 2143475-98-1

GeA-69 (GeA69)

Catalog No.: PC-60021Not For Human Use, Lab Use Only.

GeA-69 (GeA69) is a potent, selective, allosteric, cell-active PARP14 macrodomain 2 (MD2) inhibitor with Kd of 0.86 uM in ITC assays.

Packing	Price	Stock
10 mg	$48	In stock
25 mg	$88	In stock
50 mg	$128	In stock
100 mg	$198	In stock
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Biological Activity

GeA-69 (GeA69) is a potent, selective, allosteric, cell-active PARP14 macrodomain 2 (MD2) inhibitor with Kd of 0.86 uM in ITC assays.
GeA-69 displays high selectivity over other human macrodomains.
GeA-69 engages PARP14 MD2 in intact cells and prevents its localization to sites of DNA damage.

Physicochemical Properties

M.Wt	300.361
Formula	C20H16N2O
Appearance	Solid
CAS No.
Storage	Solide Powder -20 °C 12 Months; 4°C 6 Months	In Solvent -80 °C 6 Months; -20°C 6 Months
Shipping
Solubility	10 mM in DMSO
Chemical Name/SMILES	N-(2-(9H-carbazol-1-yl)phenyl)acetamide

References

1. Schuller M, et al. ACS Chem Biol. 2017 Nov 17;12(11):2866-2874.

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GeA-69 (GeA69)

Biological Activity

Physicochemical Properties

References

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