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Chemical Structure : GeA-69
CAS No.: 2143475-98-1
Catalog No.: PC-60021Not For Human Use, Lab Use Only.
GeA-69 (GeA69) is a potent, selective, allosteric, cell-active PARP14 macrodomain 2 (MD2) inhibitor with Kd of 0.86 uM in ITC assays.
| Packing | Price | Stock | Quantity |
|---|---|---|---|
| 10 mg | $48 | In stock | |
| 25 mg | $88 | In stock | |
| 50 mg | $128 | In stock | |
| 100 mg | $198 | In stock | |
| 250 mg | Get quote |
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GeA-69 (GeA69) is a potent, selective, allosteric, cell-active PARP14 macrodomain 2 (MD2) inhibitor with Kd of 0.86 uM in ITC assays.
GeA-69 displays high selectivity over other human macrodomains.
GeA-69 engages PARP14 MD2 in intact cells and prevents its localization to sites of DNA damage.
| M.Wt | 300.361 | |
| Formula | C20H16N2O | |
| Appearance | Solid | |
| Storage |
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| Solubility |
10 mM in DMSO |
|
| Chemical Name/SMILES |
N-(2-(9H-carbazol-1-yl)phenyl)acetamide |
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1. Schuller M, et al. ACS Chem Biol. 2017 Nov 17;12(11):2866-2874.
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