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Gilmelisib

Chemical Structure : Gilmelisib

CAS No.: 1845777-61-8

Gilmelisib

Catalog No.: PC-73420Not For Human Use, Lab Use Only.

Gilmelisib is a potent PI3K inhibitor with IC50 of <1 nM for PI3K p110α, exhibits antineoplastic acitvity.

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Purity & Documentation Purity: >98% (HPLC) Select Batch:

    Biological Activity

    Gilmelisib is a potent PI3K inhibitor with IC50 of <1 nM for PI3K p110α, exhibits antineoplastic acitvity.

    Physicochemical Properties

    M.Wt 547.99
    Formula C24H23ClFN5O5S
    Appearance Solid
    CAS No.
    Storage
    Solide Powder
    -20°C 12 Months; 4°C 6 Months
    In Solvent
    -80°C 6 Months; -20°C 6 Months
    Shipping
    Solubility

    10 mM in DMSO

    Chemical Name/SMILES

    2-chloro-N-(5-{3-[2-(dimethylamino)ethoxy]-4-oxo-4Hpyrido[1,2-a]pyrimidin-7-yl}-2-methoxypyridin-3-yl)-4-fluorobenzene-1-sulfonamide

    References

    1. WO2017101847 A1, compound 1

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